Ogo cabazitaxel ike Cabazitaxel emeputa

Nkọwa dị mkpirikpi:

Carbataxel bụ ihe kemịkal eji eme ọgwụ mgbochi ọrịa kansa.Carbataxel bụ ntụ ntụ na-acha ọcha ma ọ bụ na-acha ọcha nke fọrọ nke nta ka ọ bụrụ nke a na-apụghị ịsacha na mmiri, mana soluble na ethanol.Usoro mgbochi ọrịa kansa na njirimara ya yiri docetaxel, ọ bụkwa akụkụ nke ọgwụ mgbochi microtubule.Site na ijikọta ya na tubulin, kwalite mkpokọta ya n'ime microtubules, n'otu oge ahụ nwere ike igbochi ndị a achịkọtala microtubule disassembly, nke na-eme ka microtubules guzosie ike, si otú ahụ na-egbochi cell mitosis, na ọrụ interphase cell (interphasecellular function).


Nkọwa ngwaahịa

Mkpado ngwaahịa

Ozi ngwaahịa

Aha:Cabazitaxel

Nọmba CAS:183133-96-2

Usoro kemịkalụ:C45H57NO14

Nkọwapụta:99%

Agba:ọcha ma ọ bụ na-acha ọcha ntụ ntụ

Isi mmalite:Semi-synthesized na 10-DAB

Ụdị:API

Ọrụ na uru nke cabataxel

1.anti-cancer mmetụta: carbamazel nwere ike mgbochi ọrịa kansa mmetụta, nwere ike n'ụzọ dị irè igbochi uto na mgbasa nke tumor mkpụrụ ndụ, ịkpalite tumor cell apoptosis.E jiri ya tụnyere paclitaxel eke, carbataxel nwere ọrụ mgbochi ọrịa kansa dị elu yana ụdị mgbochi ọrịa cancer sara mbara.

2.safety: Cabataxel na nhazi na nhazi usoro, na-elekwasị anya n'ịkwalite nchekwa ngwaahịa na ndidi.Site n'ịgbanwe na ịkwalite nhazi kemịkal nke paclitaxel, a na-ebelata mmetụta nke mmetụta na mmeghachi omume ọjọọ.

Njirimara 3.pharmacokinetic: carbamazel nwere njirimara pharmacokinetic ka mma, nke mere na ọ ga-adị mma ma kesaa ya n'ime ahụ, ka ọ dịkwuo mma ọgwụgwọ ọgwụgwọ.

4.applicability: Enwere ike iji carbataxel na-agwọ ụdị ọrịa cancer dị iche iche, gụnyere ọrịa cancer akpa ume, ọrịa ara ara, ọrịa ovarian, ọrịa afọ, wdg. Achọpụtala ọrụ ya na nchekwa ya na ụlọ ọgwụ.

5.Scientific nkwado: Cabataxel dabeere na ọhụrụ sayensị nnyocha na nkà na ụzụ mmepe, na a pụrụ ịdabere na nkà mmụta sayensị nkwado.

Ọrụ anyị

1.Ngwaahịa:Nye elu-edu, elu-ọcha osisi wepụ, ọgwụ akụrụngwa, na ọgwụ intermediates.

2.Ọrụ nka:Mwepụta ahaziri iche nwere nkọwa pụrụ iche dị ka ihe ndị ahịa chọrọ.

Ụlọ ọrụ Hande

Bụrụ onye na-eweta akụrụngwa na ụlọ ọrụ na-eguzosi ike n'ezi ihe!

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