Usoro mmepụta maka Paclitaxel, ọgwụ a na-ejikarị eme ihe na ọgwụgwọ ọrịa cancer, bụ usoro mgbagwoju anya na ọkaibe nke na-ekpuchi ọtụtụ usoro, site na mmịpụta sitere na isi mmalite ruo n'usoro ọgwụ ikpeazụ.Akwụkwọ a ga-ewebata usoro mmepụta nkepaclitaxel, site na mmịpụta na nkwadebe.
Nzọụkwụ 1: Wepụta
PaclitaxelE sitere na ogbugbo osisi yew Pacific, Taxus pacifica.Usoro na-amalite site na nchịkọta nke ogbugbo ma na-achọkarị iji nlezianya mee ihe iji zere imebi osisi ahụ.A na-agbajikwa ihe ogbugbo ahụ anakọtara ma tinye ya na ihe mgbaze kwesịrị ekwesị, dị ka ether ma ọ bụ xylene.A na-agbaze Paclitaxel site n'ụgbụgbọ ka ọ bụrụ ihe mgbaze na nzọụkwụ a iji mepụta wepụ.
Nzọụkwụ 2: Nkewa
Mwepụta na-enwekarị ogige dị iche iche dị iche iche, ya mere paclitaxel kwesịrị ka ekewapụ ya na ogige ndị ọzọ.Nzọụkwụ a na-ejikarị chromatographic chromatography ma ọ bụ usoro nkewa ndị ọzọ kewapụ paclitaxel na ihe ndị ọzọ dabere na njirimara nke ogige ahụ.
Nzọụkwụ 3: Ọcha
Paclitaxel kewapụrụ kwesịrị ka a sachaa ya ọzọ iji wepụ adịghị ọcha ọ bụla fọdụrụ wee nweta ngwaahịa dị oke ọcha.Nke a na-agụnyekarị usoro dị ka crystallization, filtration, na recrystallization iji hụ na paclitaxel ikpeazụ bụ nke ịdị ọcha dị elu.
Nzọụkwụ 4: Synthesis (nhọrọ)
Ọ bụ ezie na e nwetara paclitaxel mbụ ahụ site na isi mmalite ndị sitere n'okike, ọtụtụ ụlọ ọrụ na-emepụta ọgwụ emepụtala ụzọ isi mee ya.Ụzọ ndị a na-eji ụzọ kemịkalụ sịntetik na-amụba mkpụrụ na ịchịkwa ma belata ịdabere na ihe ndị sitere n'okike.
Nzọụkwụ 5: Kwadebe ọgwụ ahụ
Nzọụkwụ ikpeazụ na usoro mmepụta bụ nkwadebe nke paclitaxel dị ọcha n'ime nkwadebe maka iji ọgwụ eme ihe.Nke a nwere ike ịgụnye igbasa paclitaxel n'ime ihe mgbaze kwesịrị ekwesị, dị ka mmanya ma ọ bụ ether, iji kwadebe ya n'ime nkwadebe ọgwụ.A na-akwado ụdị a na-ahụkarị ka ọ bụrụ ngwọta injectable iji hụ na dose ahụ ziri ezi.
Ejikọtara ọnụ, usoro mmepụta nkepaclitaxelbụ usoro mgbagwoju anya na ọtụtụ usoro e mere iji hụ na ịdị ọcha dị elu na njikwa nke ọgwụ ikpeazụ.Ọganihu nke usoro a dị oke mkpa maka ịnye ọgwụgwọ ọrịa cancer dị irè ma ya mere a na-emeziwanye ya mgbe niile ma na-emeziwanye ya iji gboo mkpa ahụike.
Rịba ama: A na-enweta uru na ngwa ndị nwere ike ime n'isiokwu a site na akwụkwọ ndị e bipụtara.
Yunnan Hande Biotechnology Co., Ltd. lekwasịrị anya na mmepụta nke paclitaxel ruo afọ 26, na ọ bụ onye nrụpụta onwe ya nke ọgwụ paclitaxel API nke United States FDA kwadoro, European EDQM, Australia TGA, China CFDA. , India, Japan na ndị ọzọ na-ahụ maka nchịkwa mba.Yunnan Hande paclitaxel, ntụpọ ọkọnọ, ụlọ ọrụ na-ere ahịa ozugbo, nabata ịjụ, 18187887160 (WhatsApp otu nọmba)
Oge nzipu: Ọktoba 13-2023